استاذ/

alsoud@aabu.edu.jo
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Research

Researche Title	عنــوان البحــث	Publishing Year
Design, Synthesis and Anticancer Screening of Novel Benzothiazole-Piperazine-1,2,3-Triazole Hybrids	تصميم وتحضيرومسح النشاط السرطاني....	2028
Design, synthesis and antimicrobial assessments of aminoacetylenic-piperazine nitroimidazole hybrid compounds	تصميم وتحضير....	2023
Nitroimidazoles Part 10. Synthesis, crystal structure, molecular docking, and anticancer evaluation of 4-nitroimidazole derivatives combined with piperazine moiety	نايتروايمدازول الجزء العاشر....	2023
Novel hybrid motifs of 4-nitroimidazole-piperazinyl tagged 1,2,3-triazoles: Synthesis, crystal structure, anticancer evaluations, and molecular docking study	هجين جديد....	2023
The crystal structure of 1-(N1-benzyl-2-methyl- 4-nitro-imidazol-5-yl)-4-(prop-2-yn-1-yl) piperazine, C18H21N5O2	التركيب البلوري للمركب.....	2022
Synthesis, Molecular Docking and Evaluation of Hetaryl Fragment Tagged 1H-1,2,4-Triazole Derivatives as Nematicidal Agents	تحضير .....	2021
Synthesis, anticancer activity and molecular docking studies of new 4- nitroimidazole derivatives	مشتقات نيترواميدازول: فاعليتها كمضادات للسرطان	2021
Nitroimidazoles Part 9. Synthesis, molecular docking, and anticancer evaluations of piperazine-tagged imidazole derivatives	نيترواميدازول الجزء التاسع....	2021
Green microwave versus conventional synthesis, crystal structure of 1-(4-(Benzothiazol-2- yl)piperazin-1-yl)-2-(4-phenyl-1H-1,2,3-triazol-1- yl)ethenone and HS-Analysis	الميكروويف الاخضر .....	2020
Synthesis and antibacterial activity of some new 1,2,4-triazole derivatives bearing carbohydrazide moiety	تحضير : النشاط المضاد للبكتيريا لبعض....	2020
Crystal structure of 3-(1-benzyl-2-ethyl-4-nitro-1Himidazol- 5-ylthio)-propanoic acid, C15H17N3O4S	التركيب البلوري...	2020
Real-Time and Online Monitoring of Glucose Contents by Using Molecular Imprinted Polymer-Based IDEs Sensor	الوقت الحقيقي لمراقبة ....	2019
REVIEW: "1,2,4-Triazolees : Synthetic Approaches and Pharmacological Importance". Chemistry of Heterocyclic Compounds, 2006, 42(11), 1377-1403.
"Synthesis, and Reactions of 1,5- and 1,3-Dialkyl Derivatives of (D-manno-pentitol-1-yl)-1H-1,2,4-Triazole Nucleosides Derived from 1-(Chloroalkyl)-1-Aza-2-Azoniaallene Salts". Carbohydrate Res., 1999, 318, 67-74.
"Synthesis and Antitumor Activity of Some New Phthalimide Analogues". Pharmazie, 2001, 5, 372-375.
"Conference": 2nd International Conference of Pure, Applied and Environmental Chemistry, Yarmouk University, Irbid-Jordan, 2000.
"Nitroimidazoles Part 6. Synthesis, structure and in vitro anti-HIV activity of new 5-substituted piperazinyl-4-nitroimidazole derivatives Antiviral Chemistry and Chemotherapy,2007,18(4), 191-200
"Structural Characterization of New Cd+2 Fluorescent Sensor Based on Lumazine Ligand: AM1 and ab initio studies". Spectrochimica Acta, Part A, 2007, 68(3), 728-733.
"Conference" : German Middle-East International conference,
"Nitroimidazoles, Part 1. An Unexpected Reactivity During the Cyclization of 3-(4-Amino-1-benzyl-2-ethyl-1H-imidazol-5-ylsulphanyl)-propionic Acid Methyl Ester. Synth. Commun., 2005, 35(17), 2259-2264.
"Conference" : Singapore International Chemical Conference 4 (SICC-4), Singapore, 2005
"Synthesis and Antiviral Activity of 1,5- and 1,3-Dialkyl-1,2,4-Triazoles C-Nucleosides Derived from 1-(Chloroalkyl)-1-Aza-2-Azoniaallene Salts". Nucleosides, Nucleotides, 1999, 18 (9), 1985-1994.
"Cycloadditions of 1-Aza-2-azoniaallene Cations to Alkenes" J.Chem. Soc. Perkin Trans. 1, 2000, (24), 4356-4365
"Synthesis of New 1H-1,2,4-Triazolylcoumarins and Their Antitumor and Anti-HIV Activities Chemistry of Heterocyclic Compounds, 2006,42(5),669-676.
"Conference": International Conference on Circular Dichroism, Pisa-Italy, 1997.
"Thienopyridone Nucleosides:Synthesis: Antibacterial and Antiviral Activity of 7-(Glyccosyl and D-manno-Pentitol-1-yl)-2-Chloro-4-Oxothieno?2,3-b? Pyrdine 5-Carboxylic Acids". SulfurLetters, 2000,24 (1), 13-22.
"Microwave-Assisted Synthesis And anti-HIV Activity of New Acyclic C-Nu-cleosides of 3-(D-Erythro-Tetritol-1-yl)-5-Mercapto-1,2,4-Triazoles. Part 1. Nucleosides, Nucleotides & Nucleic Acids, 2008, 27(5),469-483.
"Synthesis of Acyclic 6,7-Dihaloquinoline Nucleosides Analogues As Potential Antibacterial and Antiviral Agents". Bioorg.&Med. Chem., 2000, 8(6), 1407-1413.
"Cycloadditions of 1-Aza-2-azoniaallene Salts Derived from Coumarine and Camphor". J. prakt. Chemie, 1998, 340, 151-159.
"1H- and13C- NMR Study of some 6,7- Dihaloquinolone Nucleosides and their Derivatives". Spectroscopy Letters, 1998,31(5), 1031-1038.
"Conference" : The 8th International Symposium for Chinese Organic Chemists (ISCOC-8) The Chinese University of Hong Kong, Hong Kong-China, 2004.
"Nitroimidazole Part 3. Synthesis and anti-HIV Activity of New N-Alkyl 4-Nitroimidazoles, Bearing Benzothiazole and Benzoxazole Backbones Z.Natufrorschung (A Journal of Chemical Sciences), 2007,62b(4),523-528.
"Conference": 3rd Jordanian International Conference of Chemistry, Yarmouk University, Irbid -Jordan, 2002.
"Synthesis and Spectroscopic Analysis of Acyclic C-Nucleosides and Homo-C-Analoges from 1-(Chloroalkyl)-1-aza-2-azoniaallene Salts". Tetrahedron, 1999, 55, 751-758.
"Synthesis and anti-HIV Activity of Substituted 1,2,4-Triazolo-thiophene Derivatives". Heteroatom Chemistry, 2007, 18(4), 443-448.
"Synthesis and Antiviral Activity of 1-4(1,5-Dialkyl-1H-1,2,4-Triazol-3-yl) Methyl-Thymines". Arch. Pharm. Pharm. Med. Chem., 1999, 332, 143-144.
"Synthesis C- and N-Nucleosides from 1-Aza-2-azoniaallene and 1,3-Diaza-2-azoniaallene Salts". J. Chem. Soc., Perkin Trans.1, 1998, (5), 947-953.
"1-Aza-2-azoniaallene Salts: Reactions with Azomethines and other N-nucleophiles". J. Chem. Soc., Perkin Trans. 1, 1998, (22), 3759-3766.
"N- and C- Acyclic Thionucleoside Analogues of 1,2,3-Triazole". Heteroatom Chemistry, 2004, 15(5), 380-387.
"Conference" : The 2nd Arab Chemistry Conference, Applied Science University, Amman, Jordan, 2004.
"Reaction of 1-(Chloroalkylaza)-2-azoniaallene Salts with Alkenes. Prepation of Cyclic Azo. of (Azoalky) azonium and of Formazanium Compounds". Synthesis, 1998, 721-728.
"Conference" : The 2nd International Conference On Chemistry And Its Applications, Qatar University, Doha-Qatar, 2003.
"Quinolone Nucleoside :6,7-Dihalo-N-?- and ?-Glycosy1-1,4- Dihdro-4-Oxo-quinolone-3-Carboxylic Acids and Derivatives: Synthesis, Anti-microbial and Antiviral Activity". Nucleosides, Nucleotides, 1998, 17 (12), 2255-2266.
'Quantitative Structure-Activity Relationship (QSAR) on New Benzothiazoles derived Substituted Piperazine Derivatives' Comput. Theor. Nanoscience, accepted (2011).
"Conference" : The 7thJordanian Chemical Conference, Jordan, 2007.
"Nitroimidazoles Part 4. Synthesis and anti-HIV activity of New 5-Alkylsulfanyl and 5-(4?-Arylsulphonyl)Piperazine 4-Nitroimidazole Derivatives. Heteroatom Chemistry, 2007, 18(4), 334-340.
'In vitro anti-HIV and Antitumor Activity of New 3,6-disubstituted [1,2,4]Triazolo[3,4-b][1,3,4]Thiadiazole and Thiadiazine Analogues" Arch. Pharm. Chem. Life Sci., 2008,341(6), 365-369.
"Conference" 11th Eurasia Conference on Chemical Sciences, Dead Sea, Jordan, 2010.
"Synthesis and Biological activity of Some New 5- Sulphanyl-4-Nitroimidazole derivatives". J.Journal of Chemistry, 2007, 2(1), 11-20.
"Conference" : The 2nd International Symposium on Organic Chemistry, University of Sofia, Sofia, Bulgaria, 2008.
Conference: " 2nd North Africa Conference on Computational Physics and Chemistry, Oran-Algeria, 2010
"Amino acid derivarives Part 1. Synthesis, Antiviral and Antitumor Evaluation of New ?-Amino Acid Esters Bearing Coumarine Side Chain Acta Pharm., 2006,56(2), 175-188.
"Conference" : The 9th International Symposium for Chinese Organic Chemists(ISCOC-9), Singapore, 2006.
"Conference" : . 4th Jordanian International Conference of Chemistry, Yarmouk University, Irbid-Jordan, 2005.
"Conference" : The 5th Jordanian International Conference of Chemistry, Yarmouk University, Irbid-Jordan, 2008.
"Nitroimidazoles Part 2. Synthesis, Antiviral and Antitumor Activity of Chemistry & Biodiversity,2006, 3(5),515-526.
"Conference" : National Conference of Chemistry, Makkah, KSA, 2007.
"Phosphine-catalysed [3+2? cycloaddition of ethylbuta-2,3-dienoate and 4-quinolone-1,3-dicarboxylate" Lett. Org. Chem., 2008, 5 (1), 55-56.
"Conference" : Alexander von Humboldt Network Meeting, Giessen, Germany, 2007.
"Synthesis, Characterization and anti-HIV Activities of New Coumarine Derivatives" Z.Natufrorschung (A Journal of Chemical Sciences), 2008, 63b(1), 83-89.
"Conference" : Petra International Chemistry Conference, Jordan, 2007.
"Synthesis of 1-?-D-Glucopzranosyl-1,2,3-Triazole-4,5-Dimethyanol-4,5-bis-(Isopropylcarbamate) as Potential Antineoplastic Agent" Tetrahedron Letters, 2002, 43(22), 4021-4022.
"Synthesis and Reactions of New 3?-Deoxy-5?-Thioalkyl ?-D-Erythro-pentofuranosyl Thymines and Related Analogues". Phosphorus, Sulfur & Silicon 2003,178(12), 2551-2561.
"Conference" : Singapore International Chemical Conference 6 (SICC-6), Singapore, 2009.
"Synthesis, structure and in vitro anti-HIV activity of new pyrazole, 1,2,4-thiadiazole and 1,2,4-triazole derivatives" Phosphorus, Sulfur & Silicon, 2008, 183(10), 2621-2636.
"Nitroimidazoles Part 5. Synthesis and anti-HIV evaluation of New 5-Substituted Piperazine 4-Nitroimidazole Derivatives" Acta Pharm.,2007,57(4), 379-393.
"Thiosugar Nucleosides. Synthesis and Biological Activity of 1,3,4-Thiazole, Thiazoline and Thiourea Derivatives of 5-Thio-D-Clucose. Nucleosides, Nucleotides & Nucleic Acids, 2004, 23(11), 57-67.
"Conference" : Beyond Discipline Boundairies : Building a culture of research and education interdisciplinary Ecole National de I, Industrie Minerale, Rabat, Morocco, 2009.
"Thiosugar Nucleosides. Effect of Sulfur in Synthesis of Substituted Azido-5-Thio-D-Gluco- and Allopyranosyl-N-Nucleosides and New Isothionucleosides Derivatives Thereof". J. Carbohydr. Chem.,2005, 24(3), 237-250.
'Microwave-assisted Synthesis of Acyclic C Nucleosides From 1,2-and 1,3-Diketones" Nucleosides, Nucleotides, Nucleic Acids, 2009, 28(3), 175-183.
"DNA-Directed Alkylating Agents: Synthesis, Antitumor Activity and DNA Affinity of Bis-N, N?-Trisubstituted 1,2,4-Triazolo-piprazines". IL Farmaco, 2004, 59(1), 41-46
'Microwave-Assisted Synthesis and Antioxidant Properties of Some New 1,2,4-Triazole Derivatives J. Journal of Chemistry, 2010, 5(2), 119-129.
"Synthesis of 1,2,4-Triazole C-Nucleosides From Hydrazonyl Chloride and Nitriles Nucleosides, Nucleotides & Nucleic Acids, 2007,26(1), 37-43.
'New Sulphonamide and Carboxamide Derivatives of Acyclic C-Nucleosides of Triazolo-Thiadiazole and The Thiadiazine Analogues, Synthesis, anti-HIV and Antitumor Activity, Part 2." Nucleosides, Nucleotides & Nucleic Acids, 2008, 27(9), 1034-1044.
"A Novel C-Thionucleosides: Synthesis and Reactions of 1,5- and 1,3-Dialkyl Derivatives of (1,5-Dithio-1-Thiomethyl-D-L-Arabinopentulo-pyranosyl-1-yl)-1H-1,2,4-Triazole Nucleosides". J. Carbohydr. Chem., 2004, 23(2&3), 111-122.
"Synthesis and Anti-HIV Activity of New 6-Thioarylpyrimidines and Related Compounds" Phosphorus, Sulfur & Silicon, 2008,183(7), 1571-1583.
Synthesis and in vitro Antiproliferative Activity of new Benzothiazoles Derived Substituted Piperazine Derivatives Z. Natufrorschung (A Journal of Chemical Sciences), 2010, 65b (11), 1372-1380.
"New Glycosyl-(Carboxamide)-1,2,3-Triazole-N-1-Nucleosides: Synthesis and Anticancer Activity" Nucleosides, Nucleotides, Nucleic Acids, 2002, 21(4&5), 361-375.
"Some 2-Modified 4-Thionucleosides via Sulfur Participation and Synthesis of thio-AZT from 4-Thinofuranoid 1,2,Glycal". Phosphorus, Sulfur & Silicon, 2003, 178(7), 1199-1209.
'The Role of the Heterocycle in Bis(hydroxyphenyl)triazoles for Inhibition of 17beta-Hydroxysteroid Dehydrogenase (17beta-HSD) Type 1 and Type 2 Molecular and Cellular Endocrinology, 2009,301(1-2), 212-215.
"New AZT Analogues Having 5-Alkylsulfanyl Groups. Synthesis and Anti-HIV Activity. Nucleosides, Nucleotides & Nucleic Acids, 2007,26(3),223-230
'Synthesis and in vitro Antiproliferative Activity of New Benzothiazol Derivatives" ARKIVOC, 2008, (xv), 225-238.
"A New Class of Dihaloquinolones Bearing N-Aldehydoglycosyl carbohydr-azide, Mercaptp-1,2,4-triazole, Oxadiazoline and ?-Aminoester Precursors: Synthesis and Antimicrobial Activity". J. Brazilian Chem. Soc., 2003, 14(5), 790-796.
"Synthesis, Antitumor and Antiviral Propreties of Some 1,5-Dialkyl-1,2,4-riazoles-3-Substituted Hydrazides, 5-Mercapto-1,2,4-Triazoles, 1,3,4-Oxadiazole-2-thione and Indole. IL Farmaco, 2004, 59(10), 775-783
"Structural Assignments of 1-(?-D-Glucopyranosyl)-1,2,4-Triazoles By 1H-and 13C-NMR Study". Spectroscopy Letters, 2003, 36(5&6), 461-475.
"Synthesis of 1-?4-(1,5-Dialkyl-1H-1,2,4-Triazol-3-yl)Benzyl?-1H-Indoles and 5,6-Dihaloquinolones as Potential Antitumor candidates Org. Prepar, Proced. Intem.(OPPI), 2002, 34(6), 648-654.
"Synthesis of N-Substituted-1-Amino-2,3-Dihydro-1H -Imidazole-2-Thions N-Nucleosides and S-Glycosylated Derivatives". Nucleosides, Nucleotides, Nucleic Acids, 2003, 22(3), 299-207.
"New Benzylpiperazine Derivatives Bearing Mono- and Bis-dialkyl Substituted 1,2,4-Triazoles". Heteroatom Chemistry, 2005, 16(1), 28-32.
'Design, Synthesis, Biological Evaluation and Pharmacokinetics of Bis(hydroxyphenyl) substituted Azoles, Thiophenes, Benzenes and Aza-benzenes as Potent and selective non-steroidal inhibitors of 17beta-Hydroxysteroid dehydrogenase Type 1 (17beta-HSD1) j.Med. Chem., 2008, 51(21), 6725-6739.
"Synthesis of 3?-1,2,4-Triazolo- and 3?-1,3,4-Thiadiazolimino thmyidines HeteroatomChemistry, 2003, 14(4), 298-303.
'Novel fluorescent pH sensor based on coumarin with piperazine and imidazole substituents" Spectrochimica Acta, Part A, 2008, 71(3), 818-822.
"Synthesis and Properties of New Substituted 1,2,4-Triazoles: Potential Antitumor Agents". Bioorg.&Med. Chem., 2003, 11(8), 1701-1708.