ياسين احمد سالم السعود استاذ/ alsoud@aabu.edu.jo تحميل السيرة الذاتية orcid linkedin Google Scholar Scopus ResearchGate منصة الأردن المفتوحة للإبداع معلومات الاتصال فرعي الابحاث Researche Title عنــوان البحــث سنة النشـــر Design, Synthesis and Anticancer Screening of Novel Benzothiazole-Piperazine-1,2,3-Triazole Hybrids تصميم وتحضيرومسح النشاط السرطاني.... 2028 Design, synthesis and antimicrobial assessments of aminoacetylenic-piperazine nitroimidazole hybrid compounds تصميم وتحضير.... 2023 Nitroimidazoles Part 10. Synthesis, crystal structure, molecular docking, and anticancer evaluation of 4-nitroimidazole derivatives combined with piperazine moiety نايتروايمدازول الجزء العاشر.... 2023 Novel hybrid motifs of 4-nitroimidazole-piperazinyl tagged 1,2,3-triazoles: Synthesis, crystal structure, anticancer evaluations, and molecular docking study هجين جديد.... 2023 The crystal structure of 1-(N1-benzyl-2-methyl- 4-nitro-imidazol-5-yl)-4-(prop-2-yn-1-yl) piperazine, C18H21N5O2 التركيب البلوري للمركب..... 2022 Synthesis, Molecular Docking and Evaluation of Hetaryl Fragment Tagged 1H-1,2,4-Triazole Derivatives as Nematicidal Agents تحضير ..... 2021 Synthesis, anticancer activity and molecular docking studies of new 4- nitroimidazole derivatives مشتقات نيترواميدازول: فاعليتها كمضادات للسرطان 2021 Nitroimidazoles Part 9. Synthesis, molecular docking, and anticancer evaluations of piperazine-tagged imidazole derivatives نيترواميدازول الجزء التاسع.... 2021 Green microwave versus conventional synthesis, crystal structure of 1-(4-(Benzothiazol-2- yl)piperazin-1-yl)-2-(4-phenyl-1H-1,2,3-triazol-1- yl)ethenone and HS-Analysis الميكروويف الاخضر ..... 2020 Synthesis and antibacterial activity of some new 1,2,4-triazole derivatives bearing carbohydrazide moiety تحضير : النشاط المضاد للبكتيريا لبعض.... 2020 Crystal structure of 3-(1-benzyl-2-ethyl-4-nitro-1Himidazol- 5-ylthio)-propanoic acid, C15H17N3O4S التركيب البلوري... 2020 Real-Time and Online Monitoring of Glucose Contents by Using Molecular Imprinted Polymer-Based IDEs Sensor الوقت الحقيقي لمراقبة .... 2019 REVIEW: "1,2,4-Triazolees : Synthetic Approaches and Pharmacological Importance". Chemistry of Heterocyclic Compounds, 2006, 42(11), 1377-1403. "Synthesis, and Reactions of 1,5- and 1,3-Dialkyl Derivatives of (D-manno-pentitol-1-yl)-1H-1,2,4-Triazole Nucleosides Derived from 1-(Chloroalkyl)-1-Aza-2-Azoniaallene Salts". Carbohydrate Res., 1999, 318, 67-74. "Synthesis and Antitumor Activity of Some New Phthalimide Analogues". Pharmazie, 2001, 5, 372-375. "Conference": 2nd International Conference of Pure, Applied and Environmental Chemistry, Yarmouk University, Irbid-Jordan, 2000. "Nitroimidazoles Part 6. Synthesis, structure and in vitro anti-HIV activity of new 5-substituted piperazinyl-4-nitroimidazole derivatives Antiviral Chemistry and Chemotherapy,2007,18(4), 191-200 "Structural Characterization of New Cd+2 Fluorescent Sensor Based on Lumazine Ligand: AM1 and ab initio studies". Spectrochimica Acta, Part A, 2007, 68(3), 728-733. "Conference" : German Middle-East International conference, "Nitroimidazoles, Part 1. An Unexpected Reactivity During the Cyclization of 3-(4-Amino-1-benzyl-2-ethyl-1H-imidazol-5-ylsulphanyl)-propionic Acid Methyl Ester. Synth. Commun., 2005, 35(17), 2259-2264. "Conference" : Singapore International Chemical Conference 4 (SICC-4), Singapore, 2005 "Synthesis and Antiviral Activity of 1,5- and 1,3-Dialkyl-1,2,4-Triazoles C-Nucleosides Derived from 1-(Chloroalkyl)-1-Aza-2-Azoniaallene Salts". Nucleosides, Nucleotides, 1999, 18 (9), 1985-1994. "Cycloadditions of 1-Aza-2-azoniaallene Cations to Alkenes" J.Chem. Soc. Perkin Trans. 1, 2000, (24), 4356-4365 "Synthesis of New 1H-1,2,4-Triazolylcoumarins and Their Antitumor and Anti-HIV Activities Chemistry of Heterocyclic Compounds, 2006,42(5),669-676. "Conference": International Conference on Circular Dichroism, Pisa-Italy, 1997. "Thienopyridone Nucleosides:Synthesis: Antibacterial and Antiviral Activity of 7-(Glyccosyl and D-manno-Pentitol-1-yl)-2-Chloro-4-Oxothieno?2,3-b? Pyrdine 5-Carboxylic Acids". SulfurLetters, 2000,24 (1), 13-22. "Microwave-Assisted Synthesis And anti-HIV Activity of New Acyclic C-Nu-cleosides of 3-(D-Erythro-Tetritol-1-yl)-5-Mercapto-1,2,4-Triazoles. Part 1. Nucleosides, Nucleotides & Nucleic Acids, 2008, 27(5),469-483. "Synthesis of Acyclic 6,7-Dihaloquinoline Nucleosides Analogues As Potential Antibacterial and Antiviral Agents". Bioorg.&Med. Chem., 2000, 8(6), 1407-1413. "Cycloadditions of 1-Aza-2-azoniaallene Salts Derived from Coumarine and Camphor". J. prakt. Chemie, 1998, 340, 151-159. "1H- and13C- NMR Study of some 6,7- Dihaloquinolone Nucleosides and their Derivatives". Spectroscopy Letters, 1998,31(5), 1031-1038. "Conference" : The 8th International Symposium for Chinese Organic Chemists (ISCOC-8) The Chinese University of Hong Kong, Hong Kong-China, 2004. "Nitroimidazole Part 3. Synthesis and anti-HIV Activity of New N-Alkyl 4-Nitroimidazoles, Bearing Benzothiazole and Benzoxazole Backbones Z.Natufrorschung (A Journal of Chemical Sciences), 2007,62b(4),523-528. "Conference": 3rd Jordanian International Conference of Chemistry, Yarmouk University, Irbid -Jordan, 2002. "Synthesis and Spectroscopic Analysis of Acyclic C-Nucleosides and Homo-C-Analoges from 1-(Chloroalkyl)-1-aza-2-azoniaallene Salts". Tetrahedron, 1999, 55, 751-758. "Synthesis and anti-HIV Activity of Substituted 1,2,4-Triazolo-thiophene Derivatives". Heteroatom Chemistry, 2007, 18(4), 443-448. "Synthesis and Antiviral Activity of 1-4(1,5-Dialkyl-1H-1,2,4-Triazol-3-yl) Methyl-Thymines". Arch. Pharm. Pharm. Med. Chem., 1999, 332, 143-144. "Synthesis C- and N-Nucleosides from 1-Aza-2-azoniaallene and 1,3-Diaza-2-azoniaallene Salts". J. Chem. Soc., Perkin Trans.1, 1998, (5), 947-953. "1-Aza-2-azoniaallene Salts: Reactions with Azomethines and other N-nucleophiles". J. Chem. Soc., Perkin Trans. 1, 1998, (22), 3759-3766. "N- and C- Acyclic Thionucleoside Analogues of 1,2,3-Triazole". Heteroatom Chemistry, 2004, 15(5), 380-387. "Conference" : The 2nd Arab Chemistry Conference, Applied Science University, Amman, Jordan, 2004. "Reaction of 1-(Chloroalkylaza)-2-azoniaallene Salts with Alkenes. Prepation of Cyclic Azo. of (Azoalky) azonium and of Formazanium Compounds". Synthesis, 1998, 721-728. "Conference" : The 2nd International Conference On Chemistry And Its Applications, Qatar University, Doha-Qatar, 2003. "Quinolone Nucleoside :6,7-Dihalo-N-?- and ?-Glycosy1-1,4- Dihdro-4-Oxo-quinolone-3-Carboxylic Acids and Derivatives: Synthesis, Anti-microbial and Antiviral Activity". Nucleosides, Nucleotides, 1998, 17 (12), 2255-2266. 'Quantitative Structure-Activity Relationship (QSAR) on New Benzothiazoles derived Substituted Piperazine Derivatives' Comput. Theor. Nanoscience, accepted (2011). "Conference" : The 7thJordanian Chemical Conference, Jordan, 2007. "Nitroimidazoles Part 4. Synthesis and anti-HIV activity of New 5-Alkylsulfanyl and 5-(4?-Arylsulphonyl)Piperazine 4-Nitroimidazole Derivatives. Heteroatom Chemistry, 2007, 18(4), 334-340. 'In vitro anti-HIV and Antitumor Activity of New 3,6-disubstituted [1,2,4]Triazolo[3,4-b][1,3,4]Thiadiazole and Thiadiazine Analogues" Arch. Pharm. Chem. Life Sci., 2008,341(6), 365-369. "Conference" 11th Eurasia Conference on Chemical Sciences, Dead Sea, Jordan, 2010. "Synthesis and Biological activity of Some New 5- Sulphanyl-4-Nitroimidazole derivatives". J.Journal of Chemistry, 2007, 2(1), 11-20. "Conference" : The 2nd International Symposium on Organic Chemistry, University of Sofia, Sofia, Bulgaria, 2008. Conference: " 2nd North Africa Conference on Computational Physics and Chemistry, Oran-Algeria, 2010 "Amino acid derivarives Part 1. Synthesis, Antiviral and Antitumor Evaluation of New ?-Amino Acid Esters Bearing Coumarine Side Chain Acta Pharm., 2006,56(2), 175-188. "Conference" : The 9th International Symposium for Chinese Organic Chemists(ISCOC-9), Singapore, 2006. "Conference" : . 4th Jordanian International Conference of Chemistry, Yarmouk University, Irbid-Jordan, 2005. "Conference" : The 5th Jordanian International Conference of Chemistry, Yarmouk University, Irbid-Jordan, 2008. "Nitroimidazoles Part 2. Synthesis, Antiviral and Antitumor Activity of Chemistry & Biodiversity,2006, 3(5),515-526. "Conference" : National Conference of Chemistry, Makkah, KSA, 2007. "Phosphine-catalysed [3+2? cycloaddition of ethylbuta-2,3-dienoate and 4-quinolone-1,3-dicarboxylate" Lett. Org. Chem., 2008, 5 (1), 55-56. "Conference" : Alexander von Humboldt Network Meeting, Giessen, Germany, 2007. "Synthesis, Characterization and anti-HIV Activities of New Coumarine Derivatives" Z.Natufrorschung (A Journal of Chemical Sciences), 2008, 63b(1), 83-89. "Conference" : Petra International Chemistry Conference, Jordan, 2007. "Synthesis of 1-?-D-Glucopzranosyl-1,2,3-Triazole-4,5-Dimethyanol-4,5-bis-(Isopropylcarbamate) as Potential Antineoplastic Agent" Tetrahedron Letters, 2002, 43(22), 4021-4022. "Synthesis and Reactions of New 3?-Deoxy-5?-Thioalkyl ?-D-Erythro-pentofuranosyl Thymines and Related Analogues". Phosphorus, Sulfur & Silicon 2003,178(12), 2551-2561. "Conference" : Singapore International Chemical Conference 6 (SICC-6), Singapore, 2009. "Synthesis, structure and in vitro anti-HIV activity of new pyrazole, 1,2,4-thiadiazole and 1,2,4-triazole derivatives" Phosphorus, Sulfur & Silicon, 2008, 183(10), 2621-2636. "Nitroimidazoles Part 5. Synthesis and anti-HIV evaluation of New 5-Substituted Piperazine 4-Nitroimidazole Derivatives" Acta Pharm.,2007,57(4), 379-393. "Thiosugar Nucleosides. Synthesis and Biological Activity of 1,3,4-Thiazole, Thiazoline and Thiourea Derivatives of 5-Thio-D-Clucose. Nucleosides, Nucleotides & Nucleic Acids, 2004, 23(11), 57-67. "Conference" : Beyond Discipline Boundairies : Building a culture of research and education interdisciplinary Ecole National de I, Industrie Minerale, Rabat, Morocco, 2009. "Thiosugar Nucleosides. Effect of Sulfur in Synthesis of Substituted Azido-5-Thio-D-Gluco- and Allopyranosyl-N-Nucleosides and New Isothionucleosides Derivatives Thereof". J. Carbohydr. Chem.,2005, 24(3), 237-250. 'Microwave-assisted Synthesis of Acyclic C Nucleosides From 1,2-and 1,3-Diketones" Nucleosides, Nucleotides, Nucleic Acids, 2009, 28(3), 175-183. "DNA-Directed Alkylating Agents: Synthesis, Antitumor Activity and DNA Affinity of Bis-N, N?-Trisubstituted 1,2,4-Triazolo-piprazines". IL Farmaco, 2004, 59(1), 41-46 'Microwave-Assisted Synthesis and Antioxidant Properties of Some New 1,2,4-Triazole Derivatives J. Journal of Chemistry, 2010, 5(2), 119-129. "Synthesis of 1,2,4-Triazole C-Nucleosides From Hydrazonyl Chloride and Nitriles Nucleosides, Nucleotides & Nucleic Acids, 2007,26(1), 37-43. 'New Sulphonamide and Carboxamide Derivatives of Acyclic C-Nucleosides of Triazolo-Thiadiazole and The Thiadiazine Analogues, Synthesis, anti-HIV and Antitumor Activity, Part 2." Nucleosides, Nucleotides & Nucleic Acids, 2008, 27(9), 1034-1044. "A Novel C-Thionucleosides: Synthesis and Reactions of 1,5- and 1,3-Dialkyl Derivatives of (1,5-Dithio-1-Thiomethyl-D-L-Arabinopentulo-pyranosyl-1-yl)-1H-1,2,4-Triazole Nucleosides". J. Carbohydr. Chem., 2004, 23(2&3), 111-122. "Synthesis and Anti-HIV Activity of New 6-Thioarylpyrimidines and Related Compounds" Phosphorus, Sulfur & Silicon, 2008,183(7), 1571-1583. Synthesis and in vitro Antiproliferative Activity of new Benzothiazoles Derived Substituted Piperazine Derivatives Z. Natufrorschung (A Journal of Chemical Sciences), 2010, 65b (11), 1372-1380. "New Glycosyl-(Carboxamide)-1,2,3-Triazole-N-1-Nucleosides: Synthesis and Anticancer Activity" Nucleosides, Nucleotides, Nucleic Acids, 2002, 21(4&5), 361-375. "Some 2-Modified 4-Thionucleosides via Sulfur Participation and Synthesis of thio-AZT from 4-Thinofuranoid 1,2,Glycal". Phosphorus, Sulfur & Silicon, 2003, 178(7), 1199-1209. 'The Role of the Heterocycle in Bis(hydroxyphenyl)triazoles for Inhibition of 17beta-Hydroxysteroid Dehydrogenase (17beta-HSD) Type 1 and Type 2 Molecular and Cellular Endocrinology, 2009,301(1-2), 212-215. "New AZT Analogues Having 5-Alkylsulfanyl Groups. Synthesis and Anti-HIV Activity. Nucleosides, Nucleotides & Nucleic Acids, 2007,26(3),223-230 'Synthesis and in vitro Antiproliferative Activity of New Benzothiazol Derivatives" ARKIVOC, 2008, (xv), 225-238. "A New Class of Dihaloquinolones Bearing N-Aldehydoglycosyl carbohydr-azide, Mercaptp-1,2,4-triazole, Oxadiazoline and ?-Aminoester Precursors: Synthesis and Antimicrobial Activity". J. Brazilian Chem. Soc., 2003, 14(5), 790-796. "Synthesis, Antitumor and Antiviral Propreties of Some 1,5-Dialkyl-1,2,4-riazoles-3-Substituted Hydrazides, 5-Mercapto-1,2,4-Triazoles, 1,3,4-Oxadiazole-2-thione and Indole. IL Farmaco, 2004, 59(10), 775-783 "Structural Assignments of 1-(?-D-Glucopyranosyl)-1,2,4-Triazoles By 1H-and 13C-NMR Study". Spectroscopy Letters, 2003, 36(5&6), 461-475. "Synthesis of 1-?4-(1,5-Dialkyl-1H-1,2,4-Triazol-3-yl)Benzyl?-1H-Indoles and 5,6-Dihaloquinolones as Potential Antitumor candidates Org. Prepar, Proced. Intem.(OPPI), 2002, 34(6), 648-654. "Synthesis of N-Substituted-1-Amino-2,3-Dihydro-1H -Imidazole-2-Thions N-Nucleosides and S-Glycosylated Derivatives". Nucleosides, Nucleotides, Nucleic Acids, 2003, 22(3), 299-207. "New Benzylpiperazine Derivatives Bearing Mono- and Bis-dialkyl Substituted 1,2,4-Triazoles". Heteroatom Chemistry, 2005, 16(1), 28-32. 'Design, Synthesis, Biological Evaluation and Pharmacokinetics of Bis(hydroxyphenyl) substituted Azoles, Thiophenes, Benzenes and Aza-benzenes as Potent and selective non-steroidal inhibitors of 17beta-Hydroxysteroid dehydrogenase Type 1 (17beta-HSD1) j.Med. Chem., 2008, 51(21), 6725-6739. "Synthesis of 3?-1,2,4-Triazolo- and 3?-1,3,4-Thiadiazolimino thmyidines HeteroatomChemistry, 2003, 14(4), 298-303. 'Novel fluorescent pH sensor based on coumarin with piperazine and imidazole substituents" Spectrochimica Acta, Part A, 2008, 71(3), 818-822. "Synthesis and Properties of New Substituted 1,2,4-Triazoles: Potential Antitumor Agents". Bioorg.&Med. Chem., 2003, 11(8), 1701-1708.
